SCHEMBL29464237

SCHEMBL29464237

CS(=O)(=O)Nc1cccc(Br)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.46
ALDH1A1 P00352 4/20 0.42
KEAP1 Q14145 3/20 0.42
KDM4E B2RXH2 3/20 0.41
HPGD P15428 3/20 0.41
GLO1 Q04760 2/20 0.41
HTT P42858 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ALOX15 P16050 1/20 0.41
GRM5 P41594 1/20 0.41
HSD11B1 P28845 3/20 0.40
KCNE1 P15382 1/20 0.39
KCNA5 P22460 1/20 0.39
KCNQ1 P51787 1/20 0.39
KCND3 Q9UK17 1/20 0.39
NFE2L2 Q16236 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1333471 1.00 SCN9A (0.46) SCN9AALDH1A1KEAP1KDM4EHPGD
SCHEMBL3508304 0.80 TSHR (0.56) ALDH1A1KDM4EHPGDHTTHSD17B10
SCHEMBL8282718 0.80 ALDH1A1 (0.39) ALDH1A1KDM4EHPGDHTTHSD17B10
SCHEMBL12017942 0.78 ALDH1A1 (0.64) ALDH1A1KDM4EHPGDGLO1HSD17B10
SCHEMBL10094540 0.78 HSD11B1 (0.53) SCN9AALDH1A1KEAP1KDM4EHPGD
SCHEMBL2912664 0.77 ALDH1A1 (0.50) SCN9AALDH1A1KEAP1KDM4EHPGD
SCHEMBL14842058 0.77 HSD11B1 (0.49) SCN9AALDH1A1KEAP1KDM4EHPGD
SCHEMBL31143287 0.77 KDR (0.51) ALDH1A1KDM4EHPGDHTTHSD17B10
SCHEMBL14127502 0.77 KDR (0.51) ALDH1A1KDM4EHPGDHTTHSD17B10
SCHEMBL3006653 0.76 HSD11B1 (0.67) ALDH1A1KDM4EHPGDHTTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114258393-B Heterocyclic compounds having dual inhibitory activity of phosphatidylinositol 3-kinase delta and gamma and medical uses thereof 中国医药研究开发中心有限公司 2024-11-22 CN disclosed
CN-117295743-A Pyrrolopyrimidine derivatives as Wee-1 inhibitors 微境生物医药科技(上海)有限公司 2023-12-26 CN disclosed
CN-117222649-A Pyrrolopyrimidine derivatives, process for their preparation and their use 微境生物医药科技(上海)有限公司 2023-12-12 CN disclosed
CN-117222648-A Fused ring compounds as Wee-1 inhibitors, process for their preparation and their use 微境生物医药科技(上海)有限公司 2023-12-12 CN disclosed
CN-114258393-A Heterocyclic compound with dual phosphatidylinositol 3-kinase delta and gamma inhibitor activity and medical application thereof 中国医药研究开发中心有限公司 2022-03-29 CN disclosed