SCHEMBL2946472

SCHEMBL2946472

CCc1ccccc1-c1ccc(C=N[S@@+]([O-])C(C)(C)C)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 10/20 0.41
FEN1 P39748 10/20 0.41
TRPA1 O75762 1/20 0.35
GPR3 P46089 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
ABL1 P00519 2/20 0.33
KCNA5 P22460 1/20 0.32
BDKRB1 P46663 2/20 0.32
FFAR1 O14842 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
PTPN5 P54829 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2946461 1.00 ALOX5AP (0.41) ALOX5APFEN1TRPA1GPR3PDE3B
SCHEMBL2946467 1.00 ALOX5AP (0.41) ALOX5APFEN1TRPA1GPR3PDE3B
SCHEMBL2946464 1.00 ALOX5AP (0.41) ALOX5APFEN1TRPA1GPR3PDE3B
SCHEMBL4932481 0.77 GPR3 (0.38) GPR3
SCHEMBL4932491 0.77 GPR3 (0.38) GPR3
SCHEMBL2950123 0.76 ALOX5AP (0.50) ALOX5APFEN1TRPA1PDE3BPDE3A
SCHEMBL14809450 0.74 GRIN2D (0.45) GPR3
SCHEMBL1890675 0.74 GRIN2D (0.45) GPR3
SCHEMBL1890678 0.74 GRIN2D (0.45) GPR3
SCHEMBL14809451 0.74 GRIN2D (0.45) GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396301-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS Jerini AG (DE) 2011-12-21 EP disclosed
WO-2010091876-A2 SMALL MOLECULE BRADYKININ B1 RECEPTOR ANTAGONISTS JERINI AG (DE) 2010-08-19 WO disclosed