SCHEMBL29465610

SCHEMBL29465610

O=C(O)c1ccc2c(c1)cc(Cc1ccc(Cl)cc1C(F)(F)F)n2CCF

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.64
PPARG P37231 1/20 0.42
CCR2 P41597 2/20 0.40
MRGPRX4 Q96LA9 2/20 0.39
POLQ O75417 1/20 0.38
ABCB11 O95342 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
EPHX2 P34913 1/20 0.35
PLA2G4A P47712 1/20 0.35
LTB4R Q15722 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360545 1.00 RORC (0.64) RORCPPARGCCR2MRGPRX4POLQ
SCHEMBL28895765 0.92 RORC (0.56) RORCPPARGCCR2MRGPRX4POLQ
SCHEMBL28285110 0.92 RORC (0.55) RORCPPARGCCR2MRGPRX4POLQ
SCHEMBL28895622 0.90 RORC (0.54) RORCPPARGCCR2MRGPRX4POLQ
SCHEMBL20822477 0.89 RORC (0.52) RORCPPARGMRGPRX4EPHX2PLA2G4A
SCHEMBL28285097 0.88 RORC (0.55) RORCPPARGCCR2MRGPRX4POLQ
SCHEMBL19360544 0.88 RORC (0.65) RORCPPARGMRGPRX4POLQEPHX2
SCHEMBL29465606 0.88 RORC (0.65) RORCPPARGMRGPRX4POLQEPHX2
SCHEMBL22238330 0.88 RORC (0.51) RORCPPARGCCR2MRGPRX4POLQ
SCHEMBL22238305 0.87 RORC (0.51) RORCPPARGCCR2MRGPRX4POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109963836-B Deuterium atom substituted indole carboxamide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113227048-B Crystal form of indole carboxamide derivative and preparation method thereof 江苏恒瑞医药股份有限公司 2022-04-12 CN disclosed
CN-113365980-B Crystal form of deuterium atom substituted indole formamide derivative and preparation method thereof 江苏恒瑞医药股份有限公司 2022-04-12 CN disclosed