SCHEMBL29466348

SCHEMBL29466348

O=C(NC1CCN(C(=O)c2cccc(-c3cn4ccccc4n3)c2)CC1)c1ccnc(Nc2ccccc2)n1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.51
SMN1; SMN2 Q16637 6/20 0.51
RAB9A P51151 4/20 0.51
LMNA P02545 2/20 0.51
POLB P06746 2/20 0.51
GFER P55789 1/20 0.51
NPC1 O15118 2/20 0.48
ALDH1A1 P00352 7/20 0.48
HPGD P15428 4/20 0.48
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
MTOR P42345 1/20 0.44
SMG1 Q96Q15 1/20 0.44
HPGDS O60760 2/20 0.43
MAPK1 P28482 2/20 0.43
TP53 P04637 1/20 0.43
ATR Q13535 3/20 0.42
SYK P43405 1/20 0.42
MLLT1 Q03111 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25313050 1.00 KDM4E (0.51) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL29466302 0.88 KDM4E (0.52) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL25312201 0.88 KDM4E (0.52) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL25878981 0.88 KDM4E (0.54) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL25877628 0.85 KDM4E (0.52) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL29484624 0.85 RAB9A (0.56) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL25311588 0.85 RAB9A (0.56) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL25311960 0.83 KDM4E (0.56) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL25881212 0.81 KDM4E (0.49) KDM4ESMN1; SMN2RAB9ALMNAPOLB
SCHEMBL29466339 0.80 KDM4E (0.51) KDM4ESMN1; SMN2RAB9ALMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057932-A1 CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF 上海医药集团股份有限公司 2022-03-24 WO disclosed
WO-2022057928-A1 CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF 上海医药集团股份有限公司 2022-03-24 WO disclosed
CN-114195780-A Carbonyl heterocyclic compound and application thereof 上海医药集团股份有限公司 2022-03-18 CN disclosed
CN-114195806-A Carbonyl heterocyclic compound and application thereof 上海医药集团股份有限公司 2022-03-18 CN disclosed