SCHEMBL29468034

SCHEMBL29468034

Cc1cc(-c2ccc(F)cc2)ccc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 1/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 1/20 0.40
ACHE P22303 1/20 0.39
HSD17B1 P14061 2/20 0.38
HSD17B2 P37059 2/20 0.38
MAPK14 Q16539 1/20 0.37
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
THRB P10828 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
BCL2L1 Q07817 1/20 0.34
BAD Q92934 1/20 0.34
PGR P06401 1/20 0.34
AGXT P21549 1/20 0.34
NPC1 O15118 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22778153 1.00 TNKS2 (0.43) TNKS2ALDH1A1CYP3A4TSHRTDP1
SCHEMBL4303038 0.86 ALDH1A1 (0.55) ALDH1A1CYP3A4TSHRTDP1HSD17B1
SCHEMBL12440897 0.82 ALDH1A1 (0.46) ALDH1A1CYP3A4TSHRTDP1KDM4E
SCHEMBL306113 0.81
SCHEMBL29421562 0.81
SCHEMBL16200431 0.80 ALDH1A1 (0.48) TNKS2ALDH1A1CYP3A4TSHRTDP1
SCHEMBL458236 0.80 ALDH1A1 (0.48) TNKS2ALDH1A1CYP3A4TSHRTDP1
SCHEMBL3138385 0.79 ALDH1A1 (0.40) ALDH1A1CYP3A4KDM4EACHEMAPT
Fluoride SCHEMBL27656662 0.79 ALDH1A1 (0.40) ALDH1A1CYP3A4KDM4EACHEMAPT
Ammonia Solution, Strong SCHEMBL28164484 0.79 ALDH1A1 (0.40) ALDH1A1CYP3A4KDM4EACHEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3983392-A2 COMPOUNDS FOR THE MODULATION OF PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9 (PCSK9) SRX Cardio, LLC (US) 2022-04-20 EP disclosed
CN-114206843-A Compounds for modulating proprotein convertase subtilisin/Kexin type 9(PCSK9) SRX心脏有限责任公司 2022-03-18 CN disclosed