SCHEMBL29469487

SCHEMBL29469487

CN(C(=O)C(c1ccccc1)c1ccccc1)c1cccnc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.44
KDM4E B2RXH2 7/20 0.43
ASPH Q12797 2/20 0.43
KDM8 Q8N371 2/20 0.43
ALDH1A1 P00352 5/20 0.42
MAPT P10636 2/20 0.42
CYP3A4 P08684 2/20 0.42
TSHR P16473 2/20 0.42
ALOX15 P16050 1/20 0.42
BLM P54132 1/20 0.42
AGER Q15109 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP1A2 P05177 2/20 0.40
ATM Q13315 1/20 0.40
MYC P01106 1/20 0.39
TDP1 Q9NUW8 2/20 0.39
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29469492 0.87 L3MBTL1 (0.45) TACR1KDM4EASPHKDM8ALDH1A1
SCHEMBL28706970 0.81 TACR1 (0.42) TACR1KDM4EASPHKDM8ALDH1A1
SCHEMBL15018248 0.80 KDM4E (0.55) KDM4EASPHKDM8ALDH1A1MAPT
SCHEMBL29175509 0.79 TACR1 (0.43) TACR1KDM4EASPHKDM8ALDH1A1
SCHEMBL29469503 0.77 TACR1 (0.49) TACR1KDM4EALDH1A1MAPTTSHR
SCHEMBL29469494 0.73 KDM4C (0.49) TACR1KDM4EASPHKDM8ALDH1A1
SCHEMBL14362843 0.70 KDM4E (0.52) KDM4EASPHKDM8ALDH1A1MAPT
SCHEMBL31037167 0.70 KDM4E (0.55) KDM4EASPHKDM8ALDH1A1MAPT
SCHEMBL29469478 0.70 KMT2A (0.52) TACR1KDM4EALDH1A1MAPTTSHR
SCHEMBL22660327 0.69 TACR1 (0.40) TACR1KDM4EALDH1A1TSHRATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114206443-B Aromatic or heteroaromatic ring derivative and preparation method and application thereof 浙江海正药业股份有限公司 2024-02-09 CN disclosed
CN-114206443-A Aromatic ring or heteroaromatic ring derivative and preparation method and application thereof 浙江海正药业股份有限公司 2022-03-18 CN disclosed