SCHEMBL29469503

SCHEMBL29469503

CN(C(=O)C(c1ccccc1)c1ccccc1)c1ccccc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.49
KDM4E B2RXH2 4/20 0.48
ALDH1A1 P00352 4/20 0.48
GAA P10253 2/20 0.48
GLA P06280 1/20 0.48
HPGD P15428 1/20 0.48
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
ATM Q13315 1/20 0.48
TDP1 Q9NUW8 2/20 0.47
MAPT P10636 3/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 1/20 0.45
OPRM1 P35372 1/20 0.43
OPRL1 P41146 1/20 0.43
TSHR P16473 2/20 0.43
ALOX15 P16050 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29469478 0.84 KMT2A (0.52) TACR1KDM4EALDH1A1GAAMEN1
SCHEMBL29469494 0.82 KDM4C (0.49) TACR1KDM4EALDH1A1MEN1KMT2A
SCHEMBL1046327 0.78 ALDH1A1 (0.52) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL29469487 0.77 TACR1 (0.44) TACR1KDM4EALDH1A1GAAMEN1
SCHEMBL3930397 0.77 TSPO (0.54) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL11315869 0.77 ALDH1A1 (0.50) KDM4EALDH1A1GAAGLAHPGD
Diphenamide SCHEMBL11702462 0.76 TACR1 (0.48) TACR1KDM4EALDH1A1MEN1KMT2A
Diphenamide SCHEMBL15619425 0.75 ALDH1A1 (0.58) TACR1KDM4EALDH1A1GAAHPGD
SCHEMBL4276628 0.75 ALDH1A1 (0.49) KDM4EALDH1A1GAAGLAHPGD
Diphenamide SCHEMBL40535 0.74 KDM4E (0.48) TACR1KDM4EALDH1A1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114206443-B Aromatic or heteroaromatic ring derivative and preparation method and application thereof 浙江海正药业股份有限公司 2024-02-09 CN disclosed
CN-114206443-A Aromatic ring or heteroaromatic ring derivative and preparation method and application thereof 浙江海正药业股份有限公司 2022-03-18 CN disclosed