SCHEMBL29487253

SCHEMBL29487253

N#Cc1ccncc1-c1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.58
ALDH1A1 P00352 4/20 0.50
CYP2A6 P11509 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP11B1 P15538 2/20 0.49
CYP17A1 P05093 1/20 0.49
NPY5R Q15761 1/20 0.48
KDM4E B2RXH2 4/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
CYP2E1 P05181 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
XDH P47989 1/20 0.45
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
DHODH Q02127 1/20 0.45
PDE10A Q9Y233 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19955349 1.00 CYP11B2 (0.58) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
SCHEMBL7215513 0.87 ATR (0.50) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
SCHEMBL31264147 0.85 ESR2 (0.55) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
SCHEMBL3237467 0.85 CYP2A6 (0.58) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
SCHEMBL14856915 0.85 ESR2 (0.55) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
SCHEMBL30630392 0.85 ESR2 (0.55) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
SCHEMBL31038737 0.85 CYP2A6 (0.58) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL4596484 0.84 CYP2A6 (0.60) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4
SCHEMBL19955350 0.82 PDE3B (0.50) CYP11B2CYP2A6CYP1A2CYP11B1KDM4E
SCHEMBL7100987 0.82 CYP11B2 (0.50) CYP11B2ALDH1A1CYP2A6CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114206868-A 3- (2- (heteroaryl) -pyridin-4-yl) -5- (trifluoromethyl) -1,2, 4-oxadiazole derivatives as HDAC6 inhibitors 奥莱松基因组股份有限公司 2022-03-18 CN disclosed