SCHEMBL29487646

SCHEMBL29487646

N#CCC(=O)c1ccc(Cl)cc1Cl

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.62
MAPK1 P28482 1/20 0.62
HIF1A Q16665 1/20 0.62
ERCC5 P28715 1/20 0.56
FEN1 P39748 1/20 0.56
TSHR P16473 1/20 0.53
CASP1 P29466 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MAPT P10636 4/20 0.51
KDM4E B2RXH2 1/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
GABRA1 P14867 6/20 0.49
GABRG2 P18507 6/20 0.49
GABRB3 P28472 6/20 0.49
GABRB2 P47870 4/20 0.49
GABRB1 P18505 2/20 0.49
KCNH2 Q12809 1/20 0.48
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL954348 1.00 ALDH1A1 (0.62) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL11331688 0.86 ERCC5 (0.56) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL31515465 0.83 MAPT (0.49) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL31688020 0.83 CTSL (0.47) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL1855966 0.83 CTSL (0.47) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL4151911 0.83 KCNH2 (0.46) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL2520383 0.83 MAPT (0.49) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL12694520 0.81 MAPT (0.50) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL29403310 0.79 MAPT (0.59) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL11350806 0.79 MAPT (0.59) ALDH1A1MAPK1HIF1AERCC5FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115667253-B Compounds useful for inhibiting RET kinase 伊莱利利公司 2025-06-17 CN disclosed
CN-115667253-A Compounds useful for inhibition of RET kinase 伊莱利利公司 2023-01-31 CN disclosed
CN-109280028-B Quinoline compound and application thereof in DPP-4 enzyme inhibitor 上海医药工业研究院 2022-03-25 CN disclosed