SCHEMBL29488681

SCHEMBL29488681

CCS(=O)(=O)c1ccc(C(N)=O)nc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
GAA P10253 1/20 0.43
PSIP1 O75475 2/20 0.42
FLT4 P35916 2/20 0.41
KDR P35968 2/20 0.41
PLK4 O00444 1/20 0.41
AURKA O14965 1/20 0.41
ROCK2 O75116 1/20 0.41
CHEK2 O96017 1/20 0.41
PIM1 P11309 1/20 0.41
CDK2 P24941 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
CSNK1D P48730 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
LIMK1 P53667 1/20 0.41
CSNK2A1 P68400 1/20 0.41
CDK5 Q00535 1/20 0.41
ROCK1 Q13464 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28676474 1.00 KMT2A (0.45) KMT2AGAAPSIP1FLT4KDR
SCHEMBL15531384 0.84 NAMPT (0.51) PSIP1FLT4KDRPLK4AURKA
SCHEMBL1403612 0.84 KDM4E (0.50) KMT2APSIP1ALDH1A1KDM4E
SCHEMBL17168943 0.84 ALDH1A1 (0.40) KMT2AGAAPSIP1KIF11ALDH1A1
SCHEMBL10516843 0.83 MAPT (0.41) KMT2AGAAPSIP1KIF11ALDH1A1
SCHEMBL29488691 0.82 KMT2A (0.47) KMT2AFLT4KDRAURKAROCK2
SCHEMBL2697225 0.82 KMT2A (0.47) KMT2AFLT4KDRAURKAROCK2
SCHEMBL18248737 0.80 RORC (0.46) GAAPSIP1FLT4KDRPLK4
SCHEMBL3449352 0.79 KMT2A (0.47) KMT2AGSK3BSIRT6ALDH1A1KDM4E
SCHEMBL15530424 0.77 NAMPT (0.44) KMT2ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114230523-A Benzimidazole derivatives as modulators of ROR-gamma 生命医药有限责任公司 2022-03-25 CN disclosed