SCHEMBL29490336

SCHEMBL29490336

C=C(OCC)c1ccc2[nH]c(C3CC3)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HTR2B P41595 2/20 0.38
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
MMP2 P08253 1/20 0.36
MMP13 P45452 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29490184 0.90 NPC1 (0.51) NPC1RAB9ALMNATRPV1POLB
SCHEMBL27482373 0.78 HCRTR1 (0.46) NPC1RAB9AHRH3KMT2APOLB
SCHEMBL24233562 0.75 HTR2B (0.49) HTR2BHRH3
SCHEMBL19824770 0.74 NPC1 (0.65) NPC1RAB9ALMNATRPV1KMT2A
SCHEMBL24427996 0.73 MAPKAPK2 (0.48) NPC1RAB9AHRH3KMT2APOLB
SCHEMBL482663 0.73 ALDH1A1 (0.44) NPC1RAB9ALMNAKMT2AMAPT
SCHEMBL11364480 0.71 HTR2B (0.43) NPC1RAB9AHTR2BPOLBMAPT
SCHEMBL27526929 0.70 NPY5R (0.50) NPC1RAB9AHTR2BLMNAPKM
SCHEMBL5772605 0.69 CYP2D6 (0.52) NPC1RAB9AHTR2BMAPTHSD17B10
SCHEMBL24726102 0.69 CTNNB1 (0.53) NPC1RAB9AKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3976009-A2 BAX INHIBITORS AND USES THEREOF Case Western Reserve University (US) 2022-04-06 EP disclosed