SCHEMBL29495752

SCHEMBL29495752

CCc1nc(N)ccc1-c1cccc2ccc(-c3ccccc3)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 1/20 0.44
PARP1 P09874 1/20 0.44
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRB2 P47870 1/20 0.38
GABRA4 P48169 1/20 0.38
GABRE P78334 1/20 0.38
GABRA6 Q16445 1/20 0.38
GABRG1 Q8N1C3 1/20 0.38
GABRG3 Q99928 1/20 0.38
GABRQ Q9UN88 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22969491 1.00 ASIC3 (0.44) ASIC3PARP1PIM1PIM2GABRP
SCHEMBL29495777 0.90 NPC1 (0.39) PARP1PIM1PIM2GABRPGABRD
SCHEMBL22969279 0.90 NPC1 (0.39) PARP1PIM1PIM2GABRPGABRD
SCHEMBL22969201 0.88 CYP2A6 (0.45) PIM1PIM2DHFR
SCHEMBL29495887 0.88 CYP2A6 (0.45) PIM1PIM2DHFR
SCHEMBL22969593 0.87 MCHR1 (0.36) PIM1PIM2GABRPGABRDGABRA1
SCHEMBL29495692 0.87 MCHR1 (0.36) PIM1PIM2GABRPGABRDGABRA1
SCHEMBL22969237 0.86 MCHR1 (0.49) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29495695 0.86 MCHR1 (0.49) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22969505 0.84 TGFBR1 (0.41) PIM1PIM2MCHR1NCF1PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114269730-A 5-heteroaryl-pyridin-2-amine compounds as neuropeptide FF receptor antagonists 多曼治疗学公司 2022-04-01 CN claimed
CN-114269730-A 5-heteroaryl-pyridin-2-amine compounds as neuropeptide FF receptor antagonists 多曼治疗学公司 2022-04-01 CN disclosed