SCHEMBL29503449

SCHEMBL29503449

NC(=O)c1ccccc1-c1nnc[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.58
TYRO3 Q06418 1/20 0.58
DYRK1B Q9Y463 1/20 0.58
BCAT2 O15382 1/20 0.49
NUDT1 P36639 1/20 0.44
PARP1 P09874 7/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
BTK Q06187 1/20 0.39
METAP2 P50579 1/20 0.38
CHEK1 O14757 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1671248 0.85 KDM4E (0.50) CSNK1A1TYRO3DYRK1BNPC1RAB9A
SCHEMBL11567329 0.83 CSNK1A1 (0.40) CSNK1A1TYRO3DYRK1BBCAT2NUDT1
SCHEMBL986590 0.82 CSNK1A1 (0.47) CSNK1A1TYRO3DYRK1BBCAT2NUDT1
SCHEMBL746436 0.79 CSNK1A1 (0.38) CSNK1A1TYRO3DYRK1BBCAT2NUDT1
SCHEMBL986588 0.78 CSNK1A1 (0.46) CSNK1A1TYRO3DYRK1BBCAT2NUDT1
SCHEMBL2650295 0.73 CSNK1A1 (0.54) CSNK1A1TYRO3DYRK1BBCAT2NUDT1
SCHEMBL6825869 0.73 CSNK1A1 (1.00) CSNK1A1TYRO3DYRK1BBCAT2NUDT1
SCHEMBL20544704 0.73 BTK (0.44) CSNK1A1TYRO3DYRK1BPARP1BTK
SCHEMBL210767 0.73 BCAT2 (0.74) CSNK1A1TYRO3DYRK1BBCAT2NUDT1
SCHEMBL30514077 0.73 BCAT2 (0.74) CSNK1A1TYRO3DYRK1BBCAT2NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022198777-A1 APPLICATION OF TRIAZOLE COMPOUND IN PREPARATION OF ANTITUMOR DRUGS 苏州大学 2022-09-29 WO disclosed
CN-112999221-B Application of triazole compound in preparation of antitumor drugs 苏州大学 2022-04-12 CN disclosed
CN-112999221-B Application of triazole compound in preparation of antitumor drugs 苏州大学 2022-04-12 CN disclosed