SCHEMBL29513751

SCHEMBL29513751

[2H]C([2H])([2H])Oc1nccc(OC2CC2)c1N

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.33
MCHR1 Q99705 1/20 0.33
HTR1A P08908 2/20 0.32
ADRA2A P08913 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.31
IKBKB O14920 1/20 0.31
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30
PDE4A P27815 1/20 0.30
LOX P28300 1/20 0.30
LOXL2 Q9Y4K0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24344995 0.89 LRRK2 (0.35) LRRK2MCHR1HTR1AADRA2AADRA2B
SCHEMBL25344006 0.83 LRRK2 (0.43) LRRK2MCHR1S1PR1S1PR3PDE4A
SCHEMBL29502046 0.72 NOS2 (0.50)
SCHEMBL24344996 0.71 HCRTR1 (0.39) LRRK2HTR1AADRA2AADRA2BADRA2C
SCHEMBL29534763 0.70 LRRK2 (0.35) LRRK2HTR1AADRA2AADRA2BADRA2C
SCHEMBL24344934 0.70 LRRK2 (0.35) LRRK2HTR1AADRA2AADRA2BADRA2C
SCHEMBL3202404 0.69 IKBKB (0.45) ADRA2BHPGDSMN1; SMN2IKBKB
SCHEMBL29513590 0.69 IKBKB (0.45) ADRA2BHPGDSMN1; SMN2IKBKB
SCHEMBL29957854 0.69 SCD (0.36) MCHR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL29953312 0.66 ROCK1 (0.36) MCHR1HTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076973-A1 7-AZAINDOLE COMPOUNDS FOR INHIBITION OF BCR-ABL TYROSINE KINASES ENLIVEN THERAPEUTICS, INC. (US) 2022-04-14 WO disclosed