SCHEMBL29520454

SCHEMBL29520454

C[Si](C)(C)CCOCn1c(=O)n(COCC[Si](C)(C)C)c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.52
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
APEX1 P27695 1/20 0.40
EGFR P00533 1/20 0.38
IGF1R P08069 1/20 0.38
SRC P12931 1/20 0.38
FLT4 P35916 1/20 0.38
KDR P35968 1/20 0.38
FLT3 P36888 1/20 0.38
EPHB4 P54760 1/20 0.38
TEK Q02763 1/20 0.38
GAA P10253 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31211967 0.91 NPC1 (0.48) NPC1ALDH1A1MEN1KMT2AGAA
SCHEMBL30771170 0.89 NPC1 (0.45) NPC1ALDH1A1MEN1KMT2AAPEX1
SCHEMBL27154315 0.82 NPC1 (0.44) NPC1ALDH1A1MEN1KMT2AGAA
SCHEMBL24721138 0.81 NPC1 (0.41) NPC1EGFRIGF1RSRCFLT4
SCHEMBL30804530 0.80 TSHR (0.55) NPC1ALDH1A1L3MBTL1RAB9ASMN1; SMN2
SCHEMBL32659833 0.80 NPC1 (0.45) NPC1EGFRIGF1RSRCFLT4
SCHEMBL638070 0.80 NPC1 (0.45) NPC1ALDH1A1MEN1KMT2AAPEX1
SCHEMBL28654976 0.79 TSHR (0.56) NPC1ALDH1A1GAAL3MBTL1RAB9A
SCHEMBL30791436 0.79 CYP1A2 (0.55) NPC1ALDH1A1MEN1KMT2ARAB9A
SCHEMBL28612656 0.78 KDM4E (0.54) NPC1ALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116456985-A Pyrimidine and pyridine derivatives as HPK1 modulators and methods of use thereof 深圳市原力生命科学有限公司 2023-07-18 CN disclosed
WO-2022063140-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AS HPK1 MODULATOR AND METHODS USING SAME SHENZHEN IONOVA LIFE SCIENCE CO., LTD. (CN) 2022-03-31 WO disclosed