SCHEMBL2952133

SCHEMBL2952133

CC(C)(C)OC(=O)NCCOCCOCCNC(=O)Cc1ccc(Nc2nc(Cl)nc(Cl)n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENO1 P06733 1/20 0.44
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
MAPT P10636 1/20 0.41
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41
NPR3 P17342 2/20 0.41
IGF1R P08069 1/20 0.41
EGFR P00533 1/20 0.40
ITK Q08881 1/20 0.40
ABL1 P00519 1/20 0.40
PDGFRB P09619 1/20 0.40
SRC P12931 1/20 0.40
PDGFRA P16234 1/20 0.40
MAPK14 Q16539 1/20 0.40
KDM4E B2RXH2 2/20 0.40
GLA P06280 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18470108 0.80 ADORA2A (0.43) MEN1KMT2AMAPTNPR3ADORA2A
SCHEMBL6695129 0.78 KDM4E (0.49) MAPTEGFRITKKDM4E
SCHEMBL30679678 0.78 CA9 (0.59)
SCHEMBL16983519 0.78 CA9 (0.59)
SCHEMBL13326025 0.78 ADORA2A (0.48) MEN1KMT2AADORA2AADORA1STK17B
SCHEMBL2955788 0.77 ADORA2A (0.43) ADORA2AADORA1
SCHEMBL31478285 0.74 HDAC4 (0.43) MAPTKDM4EGLAL3MBTL1ADORA2A
SCHEMBL23345470 0.74 POLB (0.60) MEN1KMT2AMAPTCACNA1BAPBA1
SCHEMBL31681549 0.73 STK17B (0.46) MEN1KMT2AEGFRITKADORA2A
SCHEMBL17576107 0.72 NPC1 (0.51) MEN1KMT2AMAPTNPR3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7749940-B2 Facilitated forward chemical genetics using tagged triazine library NEW YORK UNIVERSITY (US) 2010-07-06 US disclosed
US-20050019831-A1 Facilitated forward chemical genetics using tagged triazine library NEW YORK UNIVERSITY (US) 2005-01-27 US disclosed
WO-2004099106-A2 FACILITATED FORWARD CHEMICAL GENETICS USING TAGGED TRIAZINE LIBRARY NEW YORK UNIVERSITY (US) 2004-11-18 WO disclosed