SCHEMBL29530701

SCHEMBL29530701

COc1cc(C(=O)N2CCN(c3ncccn3)CC2)ccc1N

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.65
HPGD P15428 1/20 0.65
KDM4E B2RXH2 3/20 0.62
SLC6A7 Q99884 9/20 0.62
LMNA P02545 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
HSD17B10 Q99714 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.56
CDK5 Q00535 1/20 0.56
CDK5R1 Q15078 1/20 0.56
TSHR P16473 1/20 0.55
USP2 O75604 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
RECQL P46063 1/20 0.54
TLR8 Q9NR97 1/20 0.53
TLR7 Q9NYK1 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15880929 0.86 ALDH1A1 (0.59) ALDH1A1HPGDLMNASMN1; SMN2HSD17B10
SCHEMBL29531076 0.81 POLB (0.63) ALDH1A1HPGDSMN1; SMN2L3MBTL1TSHR
SCHEMBL12312321 0.81 ALDH1A1 (0.54) ALDH1A1HPGDLMNASMN1; SMN2HSD17B10
SCHEMBL520418 0.81 POLB (0.63) ALDH1A1HPGDSMN1; SMN2L3MBTL1TSHR
SCHEMBL30870987 0.81 HPGD (0.64) ALDH1A1HPGDHSD17B10L3MBTL1TSHR
SCHEMBL15651739 0.81 HPGD (0.60) ALDH1A1HPGDSMN1; SMN2HSD17B10L3MBTL1
SCHEMBL30871381 0.81 HPGD (0.60) ALDH1A1HPGDSMN1; SMN2HSD17B10L3MBTL1
SCHEMBL1782181 0.81 HPGD (0.64) ALDH1A1HPGDHSD17B10L3MBTL1TSHR
SCHEMBL4418409 0.81 ALDH1A1 (0.61) ALDH1A1HPGDKDM4ESLC6A7LMNA
SCHEMBL4314298 0.81 ALDH1A1 (0.61) ALDH1A1HPGDKDM4ESLC6A7LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478539-B Novel DCLK1 inhibitor and preparation method and application thereof 中国人民解放军海军军医大学 2024-02-02 CN disclosed
CN-114478539-A Novel DCLK1 inhibitor and preparation method and application thereof 中国人民解放军海军军医大学 2022-05-13 CN disclosed