SCHEMBL29532829

SCHEMBL29532829

O=C(NCC1CCN(C(=O)OCc2ccccc2)CC1)OCc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 12/20 0.67
CYP2D6 P10635 4/20 0.66
CYP2C9 P11712 4/20 0.66
SMN1; SMN2 Q16637 3/20 0.64
NPC1 O15118 2/20 0.64
RAB9A P51151 2/20 0.64
TPSAB1 Q15661 3/20 0.63
TPSD1 Q9BZJ3 3/20 0.63
TPSG1 Q9NRR2 3/20 0.63
CYP3A4 P08684 3/20 0.62
CYP2C19 P33261 1/20 0.61
F2 P00734 1/20 0.58
PLG P00747 1/20 0.58
PRSS1 P07477 1/20 0.58
PRSS2 P07478 1/20 0.58
PRSS3 P35030 1/20 0.58
HTT P42858 1/20 0.58
F13A1 P00488 1/20 0.55
TGM2 P21980 1/20 0.55
TGM1 P22735 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1240612 0.91 TPSAB1 (0.58) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL5315258 0.90 GRIN2B (0.56) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL1241067 0.88 KDM4E (0.69) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL5351275 0.88 KDM4E (0.62) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL5366902 0.88 TPSAB1 (0.72) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL8393648 0.86 LMNA (0.58) CYP2D6CYP2C9SMN1; SMN2TPSAB1TPSD1
SCHEMBL13739493 0.86 TPSAB1 (0.53) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL13740320 0.86 TPSAB1 (0.53) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL13741073 0.86 TPSAB1 (0.53) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1
SCHEMBL4286977 0.86 GRIN2B (0.69) GRIN2BCYP2D6CYP2C9SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3468960-B1 CHEMICAL COMPOUNDS AS ATF4 PATHWAY INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2022-03-23 EP claimed
EP-3468960-B1 CHEMICAL COMPOUNDS AS ATF4 PATHWAY INHIBITORS GLAXOSMITHKLINE IP DEV LTD (GB) 2022-03-23 EP disclosed