Plx-4720

Plx-4720

SCHEMBL29537252

CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 4/20 1.00
RIPK2 O43353 2/20 1.00
RAF1 P04049 2/20 1.00
KDR P35968 2/20 1.00
MAP2K2 P36507 2/20 1.00
TGFBR2 P37173 2/20 1.00
NEK2 P51955 2/20 1.00
MAP2K1 Q02750 2/20 1.00
TNK2 Q07912 2/20 1.00
MAP2K5 Q13163 2/20 1.00
PTK6 Q13882 2/20 1.00
NEK11 Q8NG66 2/20 1.00
MAP3K20 Q9NYL2 2/20 1.00
MAP4K5 Q9Y4K4 2/20 1.00
BMPR1B O00238 1/20 1.00
PLK4 O00444 1/20 1.00
PIR O00625 1/20 1.00
AURKA O14965 1/20 1.00
DCLK1 O15075 1/20 1.00
EPHB6 O15197 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Plx-4720 SCHEMBL29392465 1.00 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2
Plx-4720 SCHEMBL133733 1.00 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL298760 0.95 BRAF (0.90) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL298198 0.94 BRAF (0.88) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL7868924 0.93 BRAF (0.88) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL298282 0.92 BRAF (0.84) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL299672 0.91 BRAF (0.83) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL298349 0.91 BRAF (0.83) BRAFRIPK2RAF1KDRMAP2K2
Vemurafenib SCHEMBL29355460 0.90 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2
SCHEMBL12891936 0.90 BRAF (1.00) BRAFRIPK2RAF1KDRMAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 71 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12522872-B2 Methods of diagnosing and treating cancer in patients having or developing resistance to a first cancer therapy DANA-FARBER CANCER INSTITUTE, INC. (US) 2026-01-13 US claimed
US-20250034652-A1 C-RAF Mutants that Confer Resistance to RAF Inhibitors DANA-FARBER CANCER INSTITUTE, INC. (US) 2025-01-30 US claimed
US-12195771-B2 Combination chemotherapy for the treatment of cancer WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2025-01-14 US claimed
US-12146196-B2 C-RAF mutants that confer resistance to RAF inhibitors DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-11-19 US claimed
US-20240093310-A1 C-RAF Mutants that Confer Resistance to RAF Inhibitors DANA-FARBER CANCER INSTITUTE, INC. (US) 2024-03-21 US claimed
US-11788151-B2 C-RAF mutants that confer resistance to RAF inhibitors DANA-FARBER CANCER INSTITUTE, INC. (US) 2023-10-17 US claimed
US-11723891-B2 Drug combinations for use in the treatment of RAS-mutant cancer UMC UTRECHT HOLDING B.V. (NL) 2023-08-15 US claimed
US-11590133-B2 Methods and compositions for treatment of BRAF mutant cancers MEMORIAL SLOAN KETTERING CANCER CENTER 2023-02-28 US claimed
CN-114761006-A Methods of treating cancer resistant to kinase inhibitors INSERM(法国国家健康医学研究院) 2022-07-15 CN claimed
US-20220195408-A1 COMBINATION CHEMOTHERAPY FOR THE TREATMENT OF CANCER WISCONSIN ALUMNI RESEARCH FOUNDATION 2022-06-23 US claimed
CN-114364798-A Combination of Dbait molecules with kinase inhibitors for the treatment of cancer 欧恩科斯欧公司 2022-04-15 CN claimed
US-11286469-B2 Combination chemotherapy for the treatment of cancer WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2022-03-29 US claimed
CN-117177975-B Pyrimido [5,4, D ] pyrimidine compounds, compositions comprising the same and uses thereof 蒙特利尔大学 2026-05-19 CN disclosed
US-20260124285-A1 PERSONALIZED CANCER VACCINES MODERNATX, INC. (US) 2026-05-07 US disclosed
US-12582609-B2 Cancer vaccines MODERNATX, INC. (US) 2026-03-24 US disclosed
EP-4648793-A1 PERSONALIZED CANCER VACCINES ModernaTX, Inc. (US) 2025-11-19 EP disclosed
US-20220125899-A1 RNA CANCER VACCINES MODERNATX, INC. (US) 2022-04-28 US disclosed
CN-114364798-A Combination of Dbait molecules with kinase inhibitors for the treatment of cancer 欧恩科斯欧公司 2022-04-15 CN disclosed
CN-114302878-A Tyrosine kinase non-receptor 1(TNK1) inhibitors and uses thereof 大日本住友制药肿瘤公司 2022-04-08 CN disclosed
US-11286469-B2 Combination chemotherapy for the treatment of cancer WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2022-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12582609-B2 Cancer vaccines RNMT, MICA, NSUN2 BRAF 1940/4885RIPK2 3996/4885RAF1 1606/4885
US-20220125899-A1 RNA CANCER VACCINES NSUN3, RNGTT, TP53 BRAF 1038/4885RIPK2 4515/4885RAF1 1594/4885
US-20260124285-A1 PERSONALIZED CANCER VACCINES PDCD1, CD274, PDCD1LG2 BRAF 210/4885RIPK2 4267/4885RAF1 1416/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.