SCHEMBL29540283

SCHEMBL29540283

c1cncc(-c2ccnc(NC3CCNCC3)n2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 5/20 0.65
MAPK8 P45983 2/20 0.57
CYP1A2 P05177 2/20 0.56
USP2 O75604 1/20 0.56
ALDH1A1 P00352 1/20 0.56
ALOX15 P16050 1/20 0.56
HIF1A Q16665 1/20 0.56
HSD17B10 Q99714 1/20 0.56
IRAK4 Q9NWZ3 1/20 0.56
ABL1 P00519 2/20 0.54
EGFR P00533 2/20 0.54
PRKCA P17252 1/20 0.54
PRKCD Q05655 1/20 0.54
CDK1 P06493 1/20 0.54
CDK4 P11802 1/20 0.54
CCNB1 P14635 1/20 0.54
CCNA2 P20248 1/20 0.54
CCND1 P24385 1/20 0.54
CDK2 P24941 1/20 0.54
CCNA1 P78396 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30565323 0.85 PRKCZ (0.52) IKBKBABL1EGFRPRKCAPRKCD
SCHEMBL29539927 0.82 IKBKB (0.67) IKBKBMAPK8ABL1EGFRPRKCA
SCHEMBL13015042 0.81 CYP1A2 (0.61) IKBKBMAPK8CYP1A2USP2ALDH1A1
SCHEMBL27739765 0.81 ABL1 (0.53) IKBKBMAPK8ABL1EGFRPRKCA
SCHEMBL27739764 0.81 HDAC8 (0.54) IKBKBMAPK8ABL1EGFRPRKCA
Hydrochloric Acid SCHEMBL3777273 0.80 CYP1A2 (0.60) IKBKBMAPK8CYP1A2USP2ALDH1A1
SCHEMBL29540237 0.80 ABL1 (0.52) IKBKBIRAK4ABL1EGFRPRKCA
SCHEMBL29541062 0.79 CYP1A2 (0.53) IKBKBMAPK8CYP1A2USP2ALDH1A1
SCHEMBL29540438 0.79 IKBKB (0.71) IKBKBMAPK8ABL1EGFRPRKCA
SCHEMBL3644540 0.79 IKBKB (0.67) IKBKBMAPK8IRAK4CDK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108276382-B Cyclin-dependent kinase inhibitor and application thereof 南京圣和药物研发有限公司 2022-10-18 CN disclosed
CN-110418789-B Derivatives of N-cycloalkyl/heterocycloalkyl-4- (imidazo [1,2-a ] pyridine) pyrimidin-2-amines as therapeutic agents 常州千红生化制药股份有限公司 2022-03-25 CN disclosed