SCHEMBL29545101

SCHEMBL29545101

O=C1NCCn2nc(-c3ccnc4[nH]ncc34)c(Cl)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 8/20 0.43
NUDT1 P36639 2/20 0.41
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
TNIK Q9UKE5 3/20 0.39
CSNK1A1 P48729 2/20 0.39
CSNK1E P49674 2/20 0.39
PIK3CA P42336 4/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CB P42338 1/20 0.37
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
MTOR P42345 3/20 0.35
BRD4 O60885 1/20 0.35
JAK2 O60674 1/20 0.34
ROCK2 O75116 1/20 0.34
PRKCA P17252 1/20 0.34
PRKCQ Q04759 1/20 0.34
PRKCD Q05655 1/20 0.34
ROCK1 Q13464 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29544753 0.83 CCNC (0.36) MAPK14
SCHEMBL31728461 0.83 CSNK1D (0.43) CSNK1DNUDT1MAPK11MAPK14TNIK
SCHEMBL31728655 0.80 CSNK1D (0.41) CSNK1DNUDT1MAPK11MAPK14TNIK
SCHEMBL29544807 0.79 HTR2C (0.33)
SCHEMBL29544554 0.78 BRD4 (0.38) CSNK1DNUDT1MAPK11MAPK14TNIK
SCHEMBL29545167 0.75 PIK3CA (0.32) CSNK1DMAPK14CSNK1A1PIK3CAMTOR
SCHEMBL29544561 0.75 MET (0.34) MAPK14PIK3CAMTOR
SCHEMBL29544960 0.75 PARP1 (0.32)
SCHEMBL29544741 0.74 CDC7 (0.36)
SCHEMBL29544520 0.73 USP7 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022072634-A1 BICYCLIC COMPOUNDS FOR USE IN THE TREATMENT CANCER SCORPION THERAPEUTICS, INC. (US) 2022-04-07 WO disclosed