SCHEMBL29549565

SCHEMBL29549565

Nc1nc(NCc2ccc3c(c2)OCO3)cc(-c2cccc(O)c2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.50
ADORA3 P0DMS8 1/20 0.50
ADORA2A P29274 1/20 0.50
ADORA1 P30542 1/20 0.50
CALM1 P0DP23 2/20 0.47
PIK3CA P42336 2/20 0.46
DYRK1A Q13627 3/20 0.45
CLK4 Q9HAZ1 3/20 0.45
VCP P55072 1/20 0.45
FYN P06241 2/20 0.45
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
GAA P10253 2/20 0.44
MAPT P10636 2/20 0.44
MAPK1 P28482 2/20 0.44
HSD17B10 Q99714 2/20 0.44
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
AURKA O14965 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22533767 1.00 BRAF (0.50) BRAFADORA3ADORA2AADORA1CALM1
SCHEMBL31456192 0.88 ADORA2A (0.57) BRAFADORA3ADORA2AADORA1DYRK1A
SCHEMBL31456247 0.88 ADORA3 (0.57) ADORA3ADORA2AADORA1DYRK1ACLK4
Hydrochloric Acid SCHEMBL30197739 0.87 TP53 (0.49) BRAFADORA3ADORA2AADORA1DYRK1A
SCHEMBL31456205 0.86 ADORA1 (0.62) ADORA3ADORA2AADORA1DYRK1ACLK4
SCHEMBL29379328 0.85 PTGDR (0.56) BRAFADORA3ADORA2AADORA1DYRK1A
SCHEMBL430891 0.85 PTGDR (0.56) BRAFADORA3ADORA2AADORA1DYRK1A
SCHEMBL31456150 0.85 HPGD (0.48) BRAFADORA3ADORA2AADORA1DYRK1A
Hydrochloric Acid SCHEMBL29549744 0.84 PTGDR (0.55) BRAFADORA3ADORA2AADORA1DYRK1A
Hydrochloric Acid SCHEMBL19668265 0.84 PTGDR (0.55) BRAFADORA3ADORA2AADORA1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3952849-A2 COMPOSITIONS AND METHODS FOR INCREASING MUSCLE MASS AND OXIDATIVE METABOLISM THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-02-16 EP disclosed