SCHEMBL29549643

SCHEMBL29549643

COC(=O)c1ccc2ncn(C3CCOC3)c2n1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.39
HCAR1 Q9BXC0 1/20 0.39
CNR2 P34972 2/20 0.38
MAP3K5 Q99683 2/20 0.36
HPGDS O60760 1/20 0.36
HTR3A P46098 4/20 0.36
ABL1 P00519 3/20 0.35
OPRM1 P35372 3/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23530232 1.00 EGFR (0.39) EGFRHCAR1CNR2MAP3K5HPGDS
SCHEMBL23530035 0.93 HCAR1 (0.45) EGFRHCAR1ALDH1A1TP53
SCHEMBL29549887 0.93 HCAR1 (0.45) EGFRHCAR1ALDH1A1TP53
SCHEMBL23554637 0.82 EGFR (0.39) EGFRCNR2MAP3K5HPGDSHTR3A
SCHEMBL23530206 0.76 IRAK4 (0.47)
SCHEMBL23529971 0.76 HCAR1 (0.40) EGFRHCAR1CNR2ABL1LRRK2
SCHEMBL29549814 0.74 ALDH1A1 (0.41) EGFRHCAR1ALDH1A1TP53LRRK2
SCHEMBL23529902 0.74 ALDH1A1 (0.41) EGFRHCAR1ALDH1A1TP53LRRK2
SCHEMBL23529998 0.74 PIM2 (0.38) CNR2ALDH1A1
SCHEMBL29549902 0.74 PIM2 (0.38) CNR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114302886-B Triazolopyridazine derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2024-03-22 CN disclosed
CN-114302886-A Triazolopyridazine derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2022-04-08 CN disclosed