SCHEMBL29558481

SCHEMBL29558481

O=C(Cl)c1cc(F)cc(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.46
CES1 P23141 3/20 0.46
TPMT P51580 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
TAS1R2 Q8TE23 1/20 0.44
HCAR1 Q9BXC0 2/20 0.39
GPR139 Q6DWJ6 1/20 0.38
GRM5 P41594 3/20 0.36
GPBAR1 Q8TDU6 1/20 0.35
IDO1 P14902 1/20 0.35
CACNA1H O95180 3/20 0.35
GRM4 Q14833 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223999 1.00 CES2 (0.46) CES2CES1TPMTTAS1R3TAS1R1
SCHEMBL2293145 0.85 CES2 (0.55) CES2CES1HCAR1
SCHEMBL114867 0.85 CES2 (0.62) CES2CES1HCAR1GRM5
SCHEMBL3358922 0.83 TPMT (0.55) CES2CES1TPMTHCAR1
SCHEMBL93282 0.83 TPMT (0.62) CES2CES1TPMTHCAR1
SCHEMBL29454778 0.82 TPMT (0.70) CES2CES1TPMTTAS1R3TAS1R1
SCHEMBL572200 0.82 TPMT (0.70) CES2CES1TPMTTAS1R3TAS1R1
Hydrochloric Acid SCHEMBL28632192 0.80 TPMT (0.59) TPMTHCAR1
SCHEMBL9631667 0.80 PARP1 (0.50) CES2CES1TPMTTAS1R3TAS1R1
SCHEMBL30463182 0.80 PARP1 (0.50) CES2CES1TPMTTAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4561563-A2 TRICYCLIC ARYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF Ensem Therapeutics, Inc. (US) 2025-06-04 EP disclosed
WO-2024067566-A1 SATURATED RING DERIVATIVE, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PHARMACEUTICAL USE THEREOF 苏州阿尔脉生物科技有限公司 2024-04-04 WO disclosed
CN-117800894-A Saturated cyclic derivative, pharmaceutical composition containing same and medical application of saturated cyclic derivative 苏州阿尔脉生物科技有限公司 2024-04-02 CN disclosed
WO-2024026129-A2 TRICYCLIC ARYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF ENSEM THERAPEUTICS, INC. (US) 2024-02-01 WO disclosed
EP-4240352-A1 T-TYPE CALCIUM CHANNEL MODULATORS AND METHODS OF USE THEREOF Praxis Precision Medicines, Inc. (US) 2023-09-13 EP disclosed
WO-2022099207-A1 T-TYPE CALCIUM CHANNEL MODULATORS AND METHODS OF USE THEREOF PRAXIS PRECISION MEDICINES, INC. (US) 2022-05-12 WO disclosed