SCHEMBL2955939

SCHEMBL2955939

CN(C)CCNc1nc(Cl)cc(N2CCCCCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
CXCR4 P61073 1/20 0.42
HRH4 Q9H3N8 1/20 0.39
RAF1 P04049 1/20 0.39
BRAF P15056 1/20 0.39
LMNA P02545 1/20 0.38
DNM2 P50570 7/20 0.38
SPIN4 Q56A73 1/20 0.37
SPIN3 Q5JUX0 1/20 0.37
SPIN2B Q9BPZ2 1/20 0.37
SPIN1 Q9Y657 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1089296 0.85 ALDH1A1 (0.61) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL1089965 0.78 CXCR4 (0.68) CXCR4HRH4DNM2
SCHEMBL1087988 0.77 CXCR4 (0.66) CXCR4HRH4DNM2
SCHEMBL9084373 0.77 HRH4 (0.49) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL26616566 0.73 HTT (0.53) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL31376309 0.73 HTT (0.53) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL12963488 0.72 RAF1 (0.56) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL9083418 0.72 KMT2A (0.54) MEN1KMT2AALDH1A1CYP1A2CYP2D6
SCHEMBL2948693 0.71 HRH4 (0.55) ALDH1A1CYP2C19HRH4DNM2
SCHEMBL1088558 0.71 CXCR4 (0.65) CXCR4HRH4DNM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120156219-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2012-06-21 US disclosed
US-20100221259-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2010-09-02 US disclosed
US-7759336-B2 Nitrogen-containing heterocyclic compounds and medicinal use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2010-07-20 US disclosed
US-20070167459-A1 Nitrogen-containing heterocyclic compounds and medicinal use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-07-19 US disclosed
EP-1571146-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2005-09-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100221259-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF CXCR4, CXCL12, CXCR3 MEN1 3648/4885KMT2A 3064/4885ALDH1A1 916/4885
US-20070167459-A1 Nitrogen-containing heterocyclic compounds and medicinal use thereof CXCR4, CXCL12, CXCR3 MEN1 3648/4885KMT2A 3064/4885ALDH1A1 916/4885
US-20120156219-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF CXCR4, CXCL12, CXCR3 MEN1 3648/4885KMT2A 3064/4885ALDH1A1 916/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.