SCHEMBL29568635

SCHEMBL29568635

COc1ccccc1Nc1ccc2c(NC(=O)c3ccc(C4CCN(C)CC4)cc3)n[nH]c2n1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 13/20 0.65
EGFR P00533 1/20 0.50
HDAC6 Q9UBN7 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
KDR P35968 2/20 0.48
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
FLT3 P36888 2/20 0.44
BRD4 O60885 1/20 0.42
BRDT Q58F21 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22551232 1.00 FGFR1 (0.65) FGFR1EGFRHDAC6HDAC3HDAC4
SCHEMBL22551202 0.89 FGFR1 (0.57) FGFR1HDAC6HDAC3HDAC4HDAC1
SCHEMBL29568745 0.88 FGFR1 (0.56) FGFR1HDAC6HDAC3HDAC4HDAC1
SCHEMBL29568146 0.88 FGFR1 (0.60) FGFR1HDAC6HDAC3HDAC4HDAC1
SCHEMBL22551239 0.88 FGFR1 (0.56) FGFR1HDAC6HDAC3HDAC4HDAC1
SCHEMBL22551204 0.88 FGFR1 (0.60) FGFR1HDAC6HDAC3HDAC4HDAC1
SCHEMBL22551168 0.86 FGFR1 (0.59) FGFR1HDAC6HDAC3HDAC4HDAC1
SCHEMBL29568126 0.86 FGFR1 (0.59) FGFR1HDAC6HDAC3HDAC4HDAC1
Acetic Acid SCHEMBL31561387 0.86 FGFR1 (0.58) FGFR1HDAC6HDAC3HDAC4HDAC1
SCHEMBL22551227 0.85 FGFR1 (0.54) FGFR1HDAC6HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3956315-B1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech Srl (IT) 2025-04-16 EP claimed
EP-3956315-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2022-02-23 EP claimed
EP-3956315-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2022-02-23 EP disclosed