SCHEMBL29574249

SCHEMBL29574249

CC(C)(C)OC(=O)N1CCN(c2cccc(OCc3ccccc3)n2)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 8/20 0.56
CKS1B P61024 2/20 0.56
SKP1 P63208 2/20 0.56
SKP2 Q13309 2/20 0.56
ACHE P22303 1/20 0.54
MAP4K4 O95819 1/20 0.52
TLR9 Q9NR96 4/20 0.51
TLR7 Q9NYK1 2/20 0.51
PRMT5 O14744 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KIT P10721 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24265269 1.00 GPR119 (0.56) GPR119CKS1BSKP1SKP2ACHE
SCHEMBL23363145 0.89 GPR119 (0.52) GPR119CKS1BSKP1SKP2ACHE
SCHEMBL29990087 0.87 GPR119 (0.51) GPR119CKS1BSKP1SKP2ACHE
SCHEMBL24670625 0.87 GPR119 (0.51) GPR119CKS1BSKP1SKP2ACHE
SCHEMBL25224739 0.85 ENPP2 (0.53) CKS1BSKP1SKP2ACHEMAP4K4
SCHEMBL3108697 0.85 HRH4 (0.46)
SCHEMBL3111974 0.83 CKS1B (0.54) GPR119CKS1BSKP1SKP2ACHE
SCHEMBL29040783 0.83 CKS1B (0.50) GPR119CKS1BSKP1SKP2ACHE
SCHEMBL31181020 0.83 CKS1B (0.54) GPR119CKS1BSKP1SKP2ACHE
SCHEMBL24337896 0.83 GPR119 (0.49) GPR119CKS1BSKP1SKP2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116507326-A Compounds as GLP-1R agonists 拓臻制药公司 2023-07-28 CN disclosed
EP-4199919-A1 COMPOUNDS AS GLP-1R AGONISTS Terns Pharmaceuticals, Inc. (US) 2023-06-28 EP disclosed
WO-2022040600-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. (US) 2022-02-24 WO disclosed