SCHEMBL29575640

SCHEMBL29575640

c1ccc2nc(Nc3ccc(-n4cccn4)cc3)ncc2c1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.58
MKNK2 Q9HBH9 1/20 0.58
SYK P43405 3/20 0.51
ROCK1 Q13464 1/20 0.46
JAK3 P52333 1/20 0.44
MAP3K5 Q99683 1/20 0.43
MAPK10 P53779 5/20 0.43
JUN P05412 2/20 0.43
MAPK8 P45983 2/20 0.43
MAP4K1 Q92918 1/20 0.42
NOTUM Q6P988 1/20 0.42
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
IGF1R P08069 1/20 0.39
STAT6 P42226 1/20 0.39
TNIK Q9UKE5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29576366 0.79 CYP11B1 (0.53) ROCK1MAP3K5MAP4K1
SCHEMBL3338544 0.77 AURKA (0.57) MKNK2SYKROCK1JAK3MAP3K5
Benzene SCHEMBL28188863 0.76 MAP3K5 (0.60) MKNK2SYKROCK1JAK3MAP3K5
SCHEMBL31381352 0.76 MAP3K5 (0.60) MKNK2SYKROCK1JAK3MAP3K5
SCHEMBL27770482 0.76 MAP3K5 (0.60) MKNK2SYKROCK1JAK3MAP3K5
SCHEMBL167891 0.76 MAP3K5 (0.60) MKNK2SYKROCK1JAK3MAP3K5
SCHEMBL3965297 0.76 JAK3 (0.53) MKNK1MKNK2SYKJAK3MAPK1
SCHEMBL5262847 0.76 CDK4 (0.73) SYKJAK3ALDH1A1
SCHEMBL3756770 0.75 MAPK10 (0.70) MKNK1MKNK2JAK3MAPK10MAPK8
SCHEMBL4573935 0.75 MAP3K5 (0.58) MKNK2SYKROCK1JAK3MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260102406-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA INC (US) 2026-04-16 US disclosed
US-12403145-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC (US) 2025-09-02 US disclosed
US-20240197752-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA INC 2024-06-20 US disclosed
US-11865120-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC. (US) 2024-01-09 US disclosed
US-20220354864-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA, INC. 2022-11-10 US disclosed
US-11304957-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC. (US) 2022-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240197752-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY DCK, ABL1, MAP4K2 MKNK1 56/4885MKNK2 47/4885SYK 721/4885
US-11865120-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 MKNK1 56/4885MKNK2 47/4885SYK 721/4885
US-12403145-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 MKNK1 56/4885MKNK2 47/4885SYK 721/4885
US-11304957-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 MKNK1 56/4885MKNK2 47/4885SYK 721/4885
US-20220354864-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY DCK, ABL1, MAP4K2 MKNK1 56/4885MKNK2 47/4885SYK 721/4885
US-20260102406-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY BRAF, TTK, MAP4K2 MKNK1 305/4885MKNK2 215/4885SYK 375/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.