SCHEMBL2958248

SCHEMBL2958248

CCOC(=O)C(=O)CC(=O)c1cccc(I)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
POLB P06746 1/20 0.54
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
GRM5 P41594 1/20 0.42
ERCC5 P28715 4/20 0.41
FEN1 P39748 4/20 0.41
MAPT P10636 1/20 0.41
GAA P10253 3/20 0.40
TP53BP1 Q12888 1/20 0.40
GPR35 Q9HC97 1/20 0.39
SYK P43405 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5482399 0.86 ERCC5 (0.46) ALDH1A1SMN1; SMN2POLBHDAC1HDAC2
SCHEMBL5621140 0.85 KMT2A (0.50) ALDH1A1HDAC1HDAC2GRM5GAA
SCHEMBL2910361 0.85 SMN1; SMN2 (0.57) ALDH1A1SMN1; SMN2POLBERCC5FEN1
SCHEMBL4689570 0.84 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2POLBGRM5MAPT
SCHEMBL29444425 0.84 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2POLBGRM5MAPT
SCHEMBL1544855 0.82 ERCC5 (0.63) ALDH1A1SMN1; SMN2POLBERCC5FEN1
SCHEMBL212542 0.82 SMN1; SMN2 (0.54) ALDH1A1SMN1; SMN2POLBHDAC1MAPT
SCHEMBL8206234 0.82 SMN1; SMN2 (0.54) ALDH1A1SMN1; SMN2POLBERCC5FEN1
SCHEMBL25011313 0.81 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2POLBERCC5FEN1
SCHEMBL7028931 0.81 KMT2A (0.56) ALDH1A1SMN1; SMN2POLBHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118908957-A Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-11-08 CN disclosed
CN-114222737-B Small molecule inhibitors of NF- κB induced kinase 詹森药业有限公司 2024-07-26 CN disclosed
CN-114222737-A Small molecule inhibitor of NF-kB induced kinase 詹森药业有限公司 2022-03-22 CN disclosed
US-7772235-B2 mGluR5 modulators ASTRAZENECA AB (SE) 2010-08-10 US disclosed
US-20080125436-A1 4-(5-{(1R)-1-[5-(3-Chlorophenyl)isoxazol-3-yl]ethoxy}-4-methyl-4H-1,2,- 4-triazol-3-yl)-1-methylpyridin-2(1H)-one; transient lower esophageal sphincter relaxations; gastroesophageal reflux disease; pain; anxiety; irritable bowel syndrome; metabotropic glutamate receptor inhibitors; peripherally acting ASTRAZENECA AB (SE) 2008-05-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080125436-A1 4-(5-{(1R)-1-[5-(3-Chlorophenyl)isoxazol-3-yl]ethoxy}-4-methyl-4H-1,2,- 4-triazol-3-yl)-1-methylpyridin-2(1H)-one; transient lower esophageal sphincter relaxations; gastroesophageal reflux disease; pain; anxiety; irritable bowel syndrome; metabotropic glutamate receptor inhibitors; peripherally acting GLRA1, GRM1, GRM5 ALDH1A1 500/4885SMN1; SMN2 1286/4885POLB 4252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.