SCHEMBL29587134

SCHEMBL29587134

CN(C)c1cccc2c1CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.54
ESR2 Q92731 1/20 0.52
NR1H2 P55055 1/20 0.51
UCHL1 P09936 1/20 0.50
SCN9A Q15858 1/20 0.48
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
ABHD6 Q9BV23 5/20 0.46
NAMPT P43490 4/20 0.44
PARP1 P09874 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
MAPT P10636 2/20 0.43
ADORA1 P30542 1/20 0.43
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2810664 1.00 MAPK1 (0.54) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL8163659 0.85 UCHL1 (0.39) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL23619623 0.84 ESR2 (0.45) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL11997414 0.83 ESR2 (0.55) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL30150268 0.83 ESR2 (0.59) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL1958196 0.83 ESR2 (0.59) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL5776971 0.83 ESR2 (0.50) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL17687111 0.83 ADORA1 (0.44) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL16730890 0.82 ESR2 (0.54) MAPK1ESR2NR1H2UCHL1SCN9A
SCHEMBL21326028 0.82 ESR2 (0.54) MAPK1ESR2NR1H2UCHL1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109863145-B Novel tetrahydroisoquinoline and tetrahydronaphthyridine compounds for the treatment and prevention of hepatitis b virus infection 豪夫迈·罗氏有限公司 2022-04-12 CN disclosed