SCHEMBL29587342

SCHEMBL29587342

C#Cc1ccc2c(c1)CCC(C(=O)NOC1CCCCO1)O2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
GSTP1 P09211 1/20 0.33
GSTM2 P28161 1/20 0.33
ACACB O00763 1/20 0.32
EPHX2 P34913 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
STS P08842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29586783 0.83 HDAC3 (0.44) NFKB1NFKB2RELACCNA2CDK2
SCHEMBL29586900 0.83 HDAC3 (0.44) NFKB1NFKB2RELACCNA2CDK2
SCHEMBL29587169 0.82 HDAC3 (0.45) CYP4F2CYP4A11NFKB1NFKB2RELA
SCHEMBL29587290 0.81 HDAC3 (0.51) CYP4F2CYP4A11NFKB1NFKB2RELA
SCHEMBL24496752 0.81 EGLN1 (0.39) CYP4F2CYP4A11HDAC3HDAC1HDAC2
SCHEMBL29586879 0.81 EGLN1 (0.39) CYP4F2CYP4A11HDAC3HDAC1HDAC2
SCHEMBL29587076 0.80 SLC6A3 (0.39) CYP4F2CYP4A11NFKB1NFKB2RELA
SCHEMBL24496697 0.78 CYP4F2 (0.40) CYP4F2CYP4A11NFKB1NFKB2RELA
SCHEMBL29586808 0.76 ITGB3 (0.41) NFKB1NFKB2RELAMEN1KMT2A
SCHEMBL24496698 0.76 CYP4F2 (0.49) CYP4F2CYP4A11NFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022120048-A1 HDAC INHIBITORS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2022-06-09 WO disclosed