SCHEMBL29588010

SCHEMBL29588010

O=C(NO)C1CCc2cc(NS(=O)(=O)c3cccc4ccccc34)ccc2O1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.50
ALDH1A1 P00352 1/20 0.49
HTT P42858 1/20 0.49
PFKFB3 Q16875 1/20 0.49
TSHR P16473 1/20 0.48
HTR6 P50406 1/20 0.44
NFKB1 P19838 5/20 0.44
NFKB2 Q00653 5/20 0.44
RELA Q04206 5/20 0.44
PGR P06401 1/20 0.43
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN5 P54829 1/20 0.43
RORA P35398 1/20 0.43
RORC P51449 1/20 0.43
NR1H2 P55055 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
GHSR Q92847 1/20 0.42
BRD4 O60885 1/20 0.42
NPY5R Q15761 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29586852 0.88 ALDH1A1 (0.47) HDAC1ALDH1A1HTTPFKFB3TSHR
SCHEMBL29587217 0.82 NFKB1 (0.52) HDAC1TSHRNFKB1NFKB2RELA
SCHEMBL4672292 0.74 HPGD (0.50) HTR6NFKB1NFKB2RELA
SCHEMBL24496758 0.72 HDAC3 (0.52) HDAC1TSHRNFKB1NFKB2RELA
SCHEMBL29587707 0.72 HDAC3 (0.52) HDAC1TSHRNFKB1NFKB2RELA
SCHEMBL24496757 0.72 HDAC3 (0.52) HDAC1TSHRNFKB1NFKB2RELA
SCHEMBL4670076 0.72 ADRB3 (0.44)
SCHEMBL14417474 0.71 HDAC1 (0.57) HDAC1ALDH1A1HTTPFKFB3TSHR
SCHEMBL29588093 0.71 NFKB1 (0.48) TSHRNFKB1NFKB2RELANPY5R
SCHEMBL24496726 0.69 MCHR1 (0.52) HDAC1HTTNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022120048-A1 HDAC INHIBITORS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2022-06-09 WO disclosed