SCHEMBL29595342

SCHEMBL29595342

COc1ccc(NC(C)=O)cc1Nc1ccnc(Nc2cc([N+](=O)[O-])c(F)cc2OC)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 8/20 0.44
AURKB Q96GD4 5/20 0.44
CDC7 O00311 1/20 0.44
IGF1R P08069 2/20 0.44
EGFR P00533 2/20 0.43
ALK Q9UM73 3/20 0.43
PRKCA P17252 1/20 0.42
ABL1 P00519 3/20 0.42
PIM1 P11309 2/20 0.42
MAPK8 P45983 2/20 0.42
GSK3B P49841 2/20 0.42
CLK4 Q9HAZ1 2/20 0.42
BCR P11274 2/20 0.42
DAPK3 O43293 1/20 0.42
JAK2 O60674 1/20 0.42
PRKD3 O94806 1/20 0.42
PAK4 O96013 1/20 0.42
RET P07949 1/20 0.42
MET P08581 1/20 0.42
FLT1 P17948 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28729729 1.00 AURKA (0.44) AURKAAURKBCDC7IGF1REGFR
SCHEMBL29594613 0.86 ALK (0.50) AURKAAURKBCDC7IGF1REGFR
SCHEMBL28728653 0.86 ALK (0.50) AURKAAURKBCDC7IGF1REGFR
SCHEMBL29594445 0.86 ALK (0.50) AURKAAURKBCDC7IGF1REGFR
SCHEMBL28729780 0.86 ALK (0.50) AURKAAURKBCDC7IGF1REGFR
SCHEMBL28729877 0.84 EGFR (0.43) AURKAAURKBCDC7IGF1REGFR
SCHEMBL29595331 0.84 ALK (0.60) IGF1REGFRALKMETMAPT
SCHEMBL28728761 0.84 ALK (0.60) IGF1REGFRALKMETMAPT
SCHEMBL30108148 0.83 ALK (0.42) AURKAAURKBCDC7IGF1REGFR
SCHEMBL19254474 0.81 EGFR (0.42) AURKAAURKBCDC7IGF1REGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394974-A Polysubstituted triaryl macrocyclic compounds and uses thereof 中国药科大学 2022-04-26 CN disclosed