SCHEMBL30108148

SCHEMBL30108148

COc1ccc(CC(N)=O)cc1Nc1ccnc(Nc2cc([N+](=O)[O-])c(F)cc2OC)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 4/20 0.42
EGFR P00533 5/20 0.42
AURKA O14965 6/20 0.41
CDK9 P50750 2/20 0.40
CCNT1 O60563 1/20 0.40
AURKB Q96GD4 3/20 0.39
CDC7 O00311 2/20 0.39
PIK3CG P48736 1/20 0.39
CAMKK2 Q96RR4 1/20 0.39
MAPK8 P45983 3/20 0.38
DAPK3 O43293 2/20 0.37
JAK2 O60674 2/20 0.37
PRKD3 O94806 2/20 0.37
PAK4 O96013 2/20 0.37
ABL1 P00519 2/20 0.37
RET P07949 2/20 0.37
IGF1R P08069 2/20 0.37
MET P08581 2/20 0.37
PIM1 P11309 2/20 0.37
FLT1 P17948 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108134 0.87 ALK (0.52) ALKEGFRAURKAAURKBCDC7
SCHEMBL30108139 0.86 ALK (0.51) ALKAURKBCDC7MAPK8DAPK3
SCHEMBL28729877 0.86 EGFR (0.43) ALKEGFRAURKACDK9CCNT1
SCHEMBL30108145 0.84 ALK (0.61) ALKIGF1RINSRLRRK2
SCHEMBL29595342 0.83 AURKA (0.44) ALKEGFRAURKACDK9AURKB
SCHEMBL28729729 0.83 AURKA (0.44) ALKEGFRAURKACDK9AURKB
SCHEMBL30108147 0.79 ALK (0.55) ALKMAPK8IGF1RMAPK9INSR
SCHEMBL30108135 0.78 ALK (0.53) ALKAURKBCDC7MAPK8DAPK3
SCHEMBL19254474 0.78 EGFR (0.42) ALKEGFRAURKACDK9CCNT1
SCHEMBL30948589 0.78 CCNT1 (0.42) ALKEGFRCDK9CCNT1AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114394974-B Polysubstituted triaryl macrocyclic compounds and uses thereof 中国药科大学 2022-12-06 CN disclosed