SCHEMBL29601443

SCHEMBL29601443

COC(=O)c1ccn(COCC[Si](C)(C)C)n1.Cc1cn(CCC[Si](C)(C)C)nc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 1/20 0.34
DGAT1 O75907 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PTGER1 P34995 1/20 0.33
KLKB1 P03952 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19926085 0.86 KMT2A (0.49) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL24537124 0.83 PTGER1 (0.39) KMT2AMEN1NPC1DGAT1PTGER1
SCHEMBL30162854 0.80 KMT2A (0.41) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL28851116 0.80 PTGER1 (0.39) KMT2AMEN1ALDH1A1PTGER1
SCHEMBL24719220 0.78 SMN1; SMN2 (0.51) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL28851114 0.78 NPC1 (0.53) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL5248123 0.77 ALDH1A1 (0.41) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL16559346 0.75 KLKB1 (0.36) KMT2AMEN1NPC1ALDH1A1DGAT1
SCHEMBL18074464 0.73 SMN1; SMN2 (0.39) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL24537117 0.73 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2ALDH1A1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115109061-A Tricyclic compounds 北京加科思新药研发有限公司 2022-09-27 CN disclosed
CN-112513041-B Tricyclic compounds 北京加科思新药研发有限公司 2022-05-10 CN disclosed