SCHEMBL29601738

SCHEMBL29601738

CCOC(=O)c1sc(Nc2cc(C)ccn2)nc1-c1ncccc1C

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 16/20 0.50
MAPT P10636 3/20 0.49
NPSR1 Q6W5P4 2/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27039803 1.00 DHODH (0.50) DHODHMAPTNPSR1KDM4ELMNA
SCHEMBL27039800 0.86 DHODH (0.53) DHODHMAPTNPSR1KDM4ELMNA
SCHEMBL19782992 0.85 DHODH (0.56) DHODHMAPTNPSR1KDM4EMEN1
SCHEMBL19782985 0.83 DHODH (0.51) DHODHMAPTNPSR1KDM4ELMNA
SCHEMBL27039903 0.81 KCNN1 (0.44) MAPTKDM4ELMNAMEN1KMT2A
SCHEMBL29601231 0.81 KCNN1 (0.44) MAPTKDM4ELMNAMEN1KMT2A
SCHEMBL19783118 0.79 DHODH (0.48) DHODHMAPTNPSR1KDM4EMEN1
SCHEMBL15993448 0.78 DHODH (0.53) DHODHMAPTNPSR1KDM4ELMNA
SCHEMBL19782993 0.78 DHODH (0.47) DHODHMAPTNPSR1KDM4EMEN1
SCHEMBL24358082 0.77 KCNN1 (0.42) MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4232449-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES Celgene Corporation (US) 2023-08-30 EP disclosed
WO-2022087326-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES CELGENE CORPORATION (US) 2022-04-28 WO disclosed