SCHEMBL29604602

SCHEMBL29604602

CN1CCC[C@@](O)(c2cccc(B3OC(C)(C)C(C)(C)O3)c2)C1=O

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.41
GRIN2A Q12879 2/20 0.41
LIPG Q9Y5X9 3/20 0.36
LPL P06858 2/20 0.36
BACE1 P56817 5/20 0.35
ROCK1 Q13464 1/20 0.33
JAK2 O60674 2/20 0.32
BTK Q06187 2/20 0.32
HSD11B1 P28845 1/20 0.32
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
OPRD1 P41143 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27129530 1.00 GRIN1 (0.41) GRIN1GRIN2ALIPGLPLBACE1
SCHEMBL26969389 1.00 GRIN1 (0.41) GRIN1GRIN2ALIPGLPLBACE1
SCHEMBL26644198 0.93 GRIN1 (0.38) GRIN1GRIN2ALIPGLPLBACE1
SCHEMBL26644195 0.93 GRIN1 (0.38) GRIN1GRIN2ALIPGLPLBACE1
SCHEMBL29605611 0.93 GRIN1 (0.38) GRIN1GRIN2ALIPGLPLBACE1
SCHEMBL29605511 0.79 GRIN1 (0.47) GRIN1GRIN2ABACE1HSD11B1ALDH1A1
SCHEMBL29604868 0.79 GRIN1 (0.47) GRIN1GRIN2ABACE1HSD11B1ALDH1A1
SCHEMBL29604635 0.77 LIPG (0.35) LIPGLPLBACE1ROCK1OPRD1
SCHEMBL27121386 0.77 LIPG (0.35) LIPGLPLBACE1ROCK1OPRD1
SCHEMBL26969399 0.77 LIPG (0.35) LIPGLPLBACE1ROCK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4244224-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE JANSSEN Pharmaceutica NV (BE) 2023-09-20 EP disclosed
WO-2022104348-A1 SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2022-05-19 WO disclosed