SCHEMBL29609014

SCHEMBL29609014

CNc1cc(Nc2cccc(OC)c2)nc(N)n1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.67
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
MAPT P10636 3/20 0.59
MAPK1 P28482 1/20 0.59
POLB P06746 3/20 0.56
RAB9A P51151 3/20 0.55
NPC1 O15118 2/20 0.55
EGFR P00533 3/20 0.53
ERBB3 P21860 2/20 0.52
ABCG2 Q9UNQ0 2/20 0.52
ABCB1 P08183 1/20 0.52
ABCC1 P33527 1/20 0.52
TP53 P04637 1/20 0.52
GALR2 O43603 2/20 0.52
GALR1 P47211 2/20 0.52
NUDT1 P36639 2/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
TNNI3K Q59H18 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28736338 1.00 ROCK1 (0.67) ROCK1MEN1KMT2AMAPTMAPK1
SCHEMBL20355235 0.86 RAB9A (0.72) ROCK1MEN1KMT2AMAPTMAPK1
SCHEMBL29609310 0.84 MAPT (0.72) ROCK1MEN1KMT2AMAPTMAPK1
SCHEMBL28736243 0.84 MAPT (0.72) ROCK1MEN1KMT2AMAPTMAPK1
SCHEMBL29610529 0.84 RAB9A (0.73) MEN1KMT2AMAPTMAPK1POLB
SCHEMBL28736336 0.84 RAB9A (0.73) MEN1KMT2AMAPTMAPK1POLB
SCHEMBL28736428 0.81 NUDT1 (0.58) MAPTPOLBRAB9ANPC1EGFR
SCHEMBL29609757 0.81 NUDT1 (0.58) MAPTPOLBRAB9ANPC1EGFR
SCHEMBL12968972 0.80 ROCK1 (1.00) ROCK1MEN1KMT2AMAPTMAPK1
SCHEMBL28736260 0.80 POLB (0.68) ROCK1MEN1KMT2AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108191774-B Heterocyclic compound, preparation method and application thereof 中国药科大学 2022-05-24 CN claimed
CN-108191774-B Heterocyclic compound, preparation method and application thereof 中国药科大学 2022-05-24 CN disclosed