SCHEMBL29610060

SCHEMBL29610060

C1=Cc2ccc(Nc3ccc4ccccc4c3)cc2CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
CYP3A4 P08684 2/20 0.50
HSD17B10 Q99714 2/20 0.50
HPGD P15428 2/20 0.50
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
EPHX2 P34913 1/20 0.38
DHFR P00374 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
SIRT3 Q9NTG7 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
SNCA P37840 1/20 0.35
MAPT P10636 5/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12887979 0.88 ALDH1A1 (0.50) ALDH1A1CYP3A4HSD17B10HPGDCYP1A2
SCHEMBL24036626 0.86 ALDH1A1 (0.44) ALDH1A1CYP3A4HSD17B10HPGDCYP1A2
SCHEMBL12956016 0.80 ALDH1A1 (0.40) ALDH1A1CYP3A4HSD17B10HPGDSNCA
SCHEMBL29609435 0.77 MAPK14 (0.51) ALDH1A1HSD17B10HPGDCYP1A2CYP2D6
Phosphoric Acid SCHEMBL30523889 0.75 ESR1 (0.39) SIRT2CA1CA2
SCHEMBL29658036 0.75 MEN1 (0.38) MEN1KMT2A
SCHEMBL325696 0.75 MEN1 (0.38) MEN1KMT2A
SCHEMBL27382283 0.74 ALDH1A1 (0.34) ALDH1A1CYP3A4HSD17B10HPGDEPHX2
SCHEMBL24296252 0.74 ALDH1A1 (0.32) ALDH1A1CYP3A4HSD17B10HPGDDHFR
SCHEMBL182655 0.74 ALDH1A1 (0.86) ALDH1A1CYP3A4HSD17B10HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022174525-A1 COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2022-08-25 WO disclosed
WO-2022174526-A1 COMPOUNDS AND MEDICAL USE THEREOF FOR COLORECTAL CANCER 中国药科大学 2022-08-25 WO disclosed
WO-2022116714-A1 COMPOUND AND MEDICAL USE THEREOF FOR NOVEL CORONAVIRUS PNEUMONIA 中国药科大学 2022-06-09 WO disclosed
CN-112920136-B Compound and medical application thereof in novel coronavirus pneumonia 中国药科大学 2022-05-03 CN disclosed