SCHEMBL29612552

SCHEMBL29612552

Nc1cc(Cl)c(Oc2ccc3ncccc3c2)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.56
CYP3A4 P08684 2/20 0.56
ALDH1A1 P00352 3/20 0.53
MAPT P10636 2/20 0.53
ATM Q13315 2/20 0.53
KDM4E B2RXH2 1/20 0.53
TP53 P04637 1/20 0.53
HSP90AA1 P07900 1/20 0.53
HSP90AB1 P08238 1/20 0.53
TSHR P16473 1/20 0.53
CASP1 P29466 1/20 0.53
HTT P42858 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HSD17B10 Q99714 1/20 0.53
CASP6 P55212 1/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
MEN1 O00255 1/20 0.48
CASP3 P42574 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23063015 1.00 PPARG (0.56) PPARGCYP3A4ALDH1A1MAPTATM
SCHEMBL23063011 0.87 PPARG (0.56) PPARGCYP3A4ALDH1A1MAPTATM
SCHEMBL9800640 0.83 MAPT (0.58) PPARGCYP3A4ALDH1A1MAPTATM
SCHEMBL3821627 0.82 ALDH1A1 (0.49) PPARGCYP3A4ALDH1A1MAPTATM
SCHEMBL633564 0.81 PPARG (0.58) PPARGCYP3A4
SCHEMBL9800721 0.80 ALDH1A1 (0.66) CYP3A4ALDH1A1MAPTATMKDM4E
SCHEMBL29612551 0.80 PPARG (0.53) PPARGCYP3A4ALDH1A1MAPTKDM4E
SCHEMBL28730677 0.80 PPARG (0.53) PPARGCYP3A4ALDH1A1MAPTKDM4E
SCHEMBL11292862 0.80 HTT (0.53) PPARGCYP3A4ALDH1A1MAPTKDM4E
SCHEMBL17164822 0.79 NPC1 (0.61) PPARGCYP3A4ALDH1A1MAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4017875-A1 THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS Terns Pharmaceuticals, Inc. (US) 2022-06-29 EP disclosed
CN-114430743-A Thyroid hormone receptor beta agonist compounds 拓臻制药公司 2022-05-03 CN disclosed