SCHEMBL29620166

SCHEMBL29620166

C(#Cc1nccc2ccccc12)c1cncnc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.50
ADORA2A P29274 1/20 0.41
PLAU P00749 2/20 0.41
CYP2A6 P11509 1/20 0.41
F12 P00748 1/20 0.41
NCF1 P14598 1/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
BACE1 P56817 1/20 0.41
ADK P55263 1/20 0.37
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
PLG P00747 1/20 0.35
EGFR P00533 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15947640 0.84 PLAU (0.54) ADORA2APLAUCYP2A6F12NCF1
SCHEMBL15940603 0.83 ADORA2A (0.54) GRM5ADORA2APLAUCYP2A6F12
Hydrochloric Acid SCHEMBL8116929 0.81 ADORA2A (0.53) GRM5ADORA2APLAUCYP2A6F12
SCHEMBL12324740 0.77 PLAU (0.49) ADORA2APLAUCYP2A6F12NCF1
SCHEMBL15947643 0.77 CYP2A6 (0.49) GRM5ADORA2APLAUCYP2A6F12
SCHEMBL17370957 0.75 CHAT (0.49) GRM5PLAUCYP2A6F12NCF1
SCHEMBL484167 0.74 S100A4 (0.51) CYP2A6ADK
SCHEMBL15947630 0.74 APP (0.44) ADORA2ACYP2A6ADKEGFR
SCHEMBL3790627 0.73 GRM5 (0.51) GRM5PLAUCYP2A6F12NCF1
SCHEMBL2431412 0.71 CYP2A6 (0.48) PLAUCYP2A6F12NCF1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220177446-A1 ALKYNE COMPOUNDS AS IRAK INHIBITORS, PREPARATION METHODS AND MEDICINAL USES THEREOF Eternity Bioscience Inc. 2022-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220177446-A1 ALKYNE COMPOUNDS AS IRAK INHIBITORS, PREPARATION METHODS AND MEDICINAL USES THEREOF IRAK2, IRAK3, IRAK4 GRM5 1155/4885ADORA2A 3455/4885PLAU 3948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.