SCHEMBL29623914

SCHEMBL29623914

COC(=O)c1nc(-c2ccccc2OC)ccc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.47
ADORA3 P0DMS8 4/20 0.47
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
ADORA1 P30542 2/20 0.44
ABL1 P00519 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
KDM6B O15054 2/20 0.43
FTO Q9C0B1 2/20 0.43
EGLN1 Q9GZT9 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
KDM2A Q9Y2K7 1/20 0.43
KDM3A Q9Y4C1 1/20 0.43
VCP P55072 1/20 0.42
PTPN1 P18031 1/20 0.42
IKBKB O14920 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HPGDS O60760 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20745147 1.00 ATR (0.47) ATRADORA3ALDH1A1HPGDADORA1
SCHEMBL20745530 0.87 ATR (0.48) ATRADORA3ALDH1A1HPGDADORA1
SCHEMBL7844018 0.79 FTO (0.58) ALDH1A1HPGDKDM6BFTOEGLN1
SCHEMBL26776167 0.79 FTO (0.40) GSK3AGSK3BKDM6BFTOEGLN1
SCHEMBL25372618 0.77 KDM4E (0.46) ATRADORA3ALDH1A1HPGDADORA1
SCHEMBL20745449 0.76 ALDH1A1 (0.47) ATRADORA3ALDH1A1HPGDADORA1
SCHEMBL1920743 0.76 PDCD1 (0.49) ADORA3ALDH1A1HPGDADORA1ABL1
SCHEMBL2463088 0.75 HSP90AA1 (0.53) ATRADORA3ALDH1A1HPGDADORA1
SCHEMBL11906808 0.74 ATR (0.53) ATRADORA3ALDH1A1HPGDABL1
SCHEMBL24658797 0.72 TP53 (0.52) ALDH1A1HPGDVCPALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3988555-A1 MACROCYCLIC MCL-1 INHIBITORS AND METHODS OF USE AbbVie Inc. (US) 2022-04-27 EP disclosed