SCHEMBL29626447

SCHEMBL29626447

COC(=O)CN(c1c(F)cc(Br)cc1OCc1ccccc1)S(=O)(=O)NC(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
MAPK1 P28482 1/20 0.43
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
KDM1A O60341 2/20 0.39
KEAP1 Q14145 5/20 0.39
NFE2L2 Q16236 5/20 0.39
PTPN1 P18031 3/20 0.39
PTPN2 P17706 2/20 0.39
PTPN6 P29350 2/20 0.39
PTPRF P10586 1/20 0.37
PTPN11 Q06124 1/20 0.37
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
CYP2C9 P11712 1/20 0.36
PTGER1 P34995 1/20 0.36
AAK1 Q2M2I8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2888862 1.00 ALDH1A1 (0.43) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL28710605 0.93 KEAP1 (0.46) CA12CA1CA7CA14KDM1A
SCHEMBL2893397 0.91 ALDH1A1 (0.44) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL2889117 0.88 ALDH1A1 (0.45) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL23540005 0.86 ALDH1A1 (0.43) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL30026722 0.86 ALDH1A1 (0.43) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL31277365 0.86 ALDH1A1 (0.43) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL30027118 0.86 ALDH1A1 (0.43) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL23540523 0.86 ALDH1A1 (0.43) ALDH1A1MAPK1CA12CA1CA7
SCHEMBL2892950 0.83 ALDH1A1 (0.48) ALDH1A1MAPK1KDM1AKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116829555-A Protein tyrosine phosphatase inhibitors and methods of use thereof 卡里科生命科学有限责任公司 2023-09-29 CN disclosed
EP-4211122-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Calico Life Sciences LLC (US) 2023-07-19 EP disclosed
CN-116332873-A Protein tyrosine phosphatase inhibitors and methods of use thereof 卡里科生命科学有限责任公司 2023-06-27 CN disclosed
WO-2022056281-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF CALICO LIFE SCIENCES LLC (US) 2022-03-17 WO disclosed