SCHEMBL29627907

SCHEMBL29627907

CCCCOC(=O)n1ncc2cc(C#Cc3ccnc(-c4ccnc(Cl)n4)n3)ccc21

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.36
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
SLC22A12 Q96S37 1/20 0.32
ACACB O00763 2/20 0.31
PLA2G4A P47712 1/20 0.31
MAPT P10636 1/20 0.31
HSP90AB1 P08238 1/20 0.31
HAO1 Q9UJM8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29627860 0.85 ROCK2 (0.38) FFAR1SLC22A12HSP90AB1HAO1
SCHEMBL29640830 0.85 ROCK2 (0.38) FFAR1SLC22A12HSP90AB1HAO1
SCHEMBL25195353 0.85 ROCK2 (0.38) FFAR1SLC22A12HSP90AB1HAO1
SCHEMBL25207952 0.83 FFAR1 (0.42) FFAR1KMT2ASLC22A12MAPTHSP90AB1
SCHEMBL29627914 0.81 FFAR1 (0.34) FFAR1PLA2G4A
SCHEMBL29627918 0.79
SCHEMBL29576192 0.76 KMT2A (0.37) ALDH1A1KMT2ASLC22A12PLA2G4AMAPT
SCHEMBL26290157 0.72 ROCK2 (0.36) ACACB
SCHEMBL26289761 0.72 ROCK2 (0.42) ACACB
SCHEMBL26289720 0.71 ROCK2 (0.38) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4003340-A2 ETHYNYLHETEROCYCLES AS RHO-ASSOCIATED COILED-COIL KINASE (ROCK) INHIBITORS Angion Biomedica Corp. (US) 2022-06-01 EP disclosed