Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL29627930

O=C(COc1ccc2c(c1)CN(c1nccc(-c3nccc(C#Cc4ccc5[nH]ncc5c4)n3)n1)C2)NC1CC1.O=C(O)C(F)(F)F

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 20/20 0.44
ROCK1 Q13464 14/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29640775 0.87 ROCK2 (0.48) ROCK2ROCK1
Trifluoroacetic Acid SCHEMBL29627947 0.83 ROCK2 (0.42) ROCK2ROCK1
SCHEMBL29640766 0.83 ROCK2 (0.44) ROCK2ROCK1
SCHEMBL29640440 0.82 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL29627927 0.81 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL29627828 0.80 ROCK2 (0.58) ROCK2ROCK1
SCHEMBL29908253 0.79 ROCK2 (0.49) ROCK2ROCK1
SCHEMBL29627716 0.78 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL29627964 0.78 ROCK2 (0.46) ROCK2ROCK1
SCHEMBL29627761 0.77 ROCK2 (0.56) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4003340-A2 ETHYNYLHETEROCYCLES AS RHO-ASSOCIATED COILED-COIL KINASE (ROCK) INHIBITORS Angion Biomedica Corp. (US) 2022-06-01 EP disclosed
CN-114502163-A Ethynylheterocycles as RHO-related coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2022-05-13 CN disclosed