SCHEMBL29629440

SCHEMBL29629440

Oc1cc(I)c2ccnc-2[nH]1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 2/20 0.33
USP2 O75604 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 2/20 0.33
HSP90AA1 P07900 2/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 2/20 0.33
SLC6A2 P23975 2/20 0.33
MAPK1 P28482 2/20 0.33
HTT P42858 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HIF1A Q16665 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27325562 0.69 KDM4E (0.30) KDM4EALDH1A1HPGDMAPK1HSD17B10
SCHEMBL7878556 0.63 NUDT1 (0.37) KDM4EMEN1ALDH1A1MAPK1KMT2A
SCHEMBL29629433 0.63 COMT (0.39) KDM4EALDH1A1LMNAHPGDALOX15
SCHEMBL3126519 0.61 PRKCI (0.33) KDM4EALDH1A1HPGDMAPK1PDE3A
SCHEMBL7878810 0.58 CDC7 (0.45) MAPK1EGFRMAPK14CYP1A2
SCHEMBL1188205 0.57 CSNK2A2 (0.30)
SCHEMBL19998636 0.56 PRKCI (0.34) KDM4EMEN1ALDH1A1HPGDMAPK1
Hydrochloric Acid SCHEMBL28275525 0.56 ALDH1A1 (0.42) KDM4EMEN1ALDH1A1HPGDMAPK1
SCHEMBL1504317 0.56 IDO1 (0.48) LMNASMN1; SMN2MAPK14HSD17B10
SCHEMBL28654223 0.56 NISCH (0.50) KDM4EMEN1ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3994138-A1 ESTROGEN-RELATED RECEPTOR ALPHA (ERRalpha) MODULATORS Lead Pharma Holding B.V. (NL) 2022-05-11 EP disclosed