SCHEMBL29631019

SCHEMBL29631019

O=C(O)c1cnc(Cc2ccccc2F)s1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
ABL1 P00519 1/20 0.44
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
PTGER1 P34995 1/20 0.42
VNN1 O95497 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HCAR2 Q8TDS4 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
DGAT1 O75907 1/20 0.39
BRS3 P32247 1/20 0.39
PKM P14618 1/20 0.39
MAPT P10636 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
GLS O94925 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20894099 1.00 NPC1 (0.45) NPC1RAB9AABL1MEN1KMT2A
SCHEMBL11782006 0.80 PTGER1 (0.46) NPC1RAB9AABL1MEN1KMT2A
SCHEMBL31482211 0.76 VNN1 (0.53) NPC1RAB9AABL1MEN1KMT2A
SCHEMBL8345339 0.76 HCAR2 (0.42) NPC1RAB9AABL1MEN1KMT2A
SCHEMBL29846096 0.74 HCAR2 (0.48) PTGER1HCAR2DGAT1BRS3GLS
SCHEMBL28854654 0.74 HCAR2 (0.48) PTGER1HCAR2DGAT1BRS3GLS
SCHEMBL9642872 0.72 HCAR2 (0.52) ALDH1A1HCAR2KDM4E
SCHEMBL6662966 0.72 HDAC1 (0.49) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL17967192 0.72 DAO (0.50) NPC1RAB9AALDH1A1HCAR2KDM4E
SCHEMBL5215834 0.72 KDM4E (0.42) NPC1RAB9AMEN1KMT2APTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563094-B (hetero) aryl-substituted piperidinyl derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2022-03-18 CN disclosed