SCHEMBL29633886

SCHEMBL29633886

COc1ccc(CCC(C(=O)O)N(C)C(=O)OCC2c3ccccc3-c3ccccc32)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 2/20 0.39
FABP5 Q01469 2/20 0.38
MDM4 O15151 2/20 0.36
TP53 P04637 2/20 0.36
EPHX2 P34913 1/20 0.35
FFAR1 O14842 2/20 0.35
P2RX7 Q99572 1/20 0.35
FABP7 O15540 1/20 0.34
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
KIF11 P52732 1/20 0.34
ALDH1A1 P00352 2/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
POLB P06746 1/20 0.33
NR1H3 Q13133 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PIK3CG P48736 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29633876 0.92 FABP5 (0.38) MDM2FABP5MDM4TP53EPHX2
SCHEMBL31688678 0.91 FABP5 (0.42) MDM2FABP5ALDH1A1POLBKDM4E
SCHEMBL29633996 0.89 FABP5 (0.34) MDM2FABP5MDM4TP53EPHX2
SCHEMBL29633788 0.88 FABP5 (0.38) MDM2FABP5MDM4TP53EPHX2
SCHEMBL31370296 0.88 FABP5 (0.38) MDM2FABP5MDM4TP53EPHX2
SCHEMBL29633900 0.87 MDM2 (0.38) MDM2FABP5MDM4TP53EPHX2
SCHEMBL29633922 0.85 MDM2 (0.43) MDM2FABP5FFAR1FABP7ALDH1A1
SCHEMBL31369914 0.85 MDM2 (0.43) MDM2FABP5FFAR1FABP7ALDH1A1
SCHEMBL31369777 0.85 FABP5 (0.39) MDM2FABP5EPHX2
SCHEMBL29634040 0.85 FABP5 (0.39) MDM2FABP5EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240376044-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 2024-11-14 US disclosed
US-12071396-B2 Method for preparing aromatic amino acid derivative CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2024-08-27 US disclosed
US-20220144762-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2022-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240376044-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE DDC, AADAT, TYR MDM2 223/4885FABP5 608/4885MDM4 381/4885
US-20220144762-A1 METHOD FOR PREPARING AROMATIC AMINO ACID DERIVATIVE DDC, AADAT, TYR MDM2 223/4885FABP5 608/4885MDM4 381/4885
US-12071396-B2 Method for preparing aromatic amino acid derivative DDC, AADAT, TYR MDM2 223/4885FABP5 608/4885MDM4 381/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.