SCHEMBL29634495

SCHEMBL29634495

COCCNC(=O)c1cccnc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.76
MEN1 O00255 5/20 0.76
CYP3A4 P08684 2/20 0.76
CYP1A2 P05177 1/20 0.76
CYP2C9 P11712 2/20 0.68
CYP2C19 P33261 2/20 0.68
ALOX15 P16050 1/20 0.68
HSD17B10 Q99714 1/20 0.68
USP2 O75604 1/20 0.67
THRB P10828 1/20 0.64
ALDH1A1 P00352 3/20 0.64
MAPT P10636 1/20 0.64
PKM P14618 1/20 0.64
TDP1 Q9NUW8 1/20 0.64
SMN1; SMN2 Q16637 4/20 0.63
LMNA P02545 2/20 0.63
POLB P06746 1/20 0.63
NPC1 O15118 2/20 0.62
RAB9A P51151 2/20 0.62
GAA P10253 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1116738 1.00 KMT2A (0.76) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL5555262 0.91 GAA (0.74) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL25328235 0.87 THRB (0.77) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL4143110 0.87 KMT2A (1.00) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL7892909 0.86 KMT2A (0.67) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL19591887 0.85 KMT2A (0.73) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL20254508 0.85 KMT2A (0.69) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL16448998 0.85 KMT2A (0.69) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL10886794 0.85 HDAC1 (0.70) KMT2AMEN1CYP3A4CYP1A2CYP2C9
SCHEMBL29447171 0.85 USP2 (0.80) KMT2AMEN1CYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107344936-B Triazolopyridazine derivative, preparation method, pharmaceutical composition and application thereof 上海赛默罗生物科技有限公司 2022-06-03 CN disclosed