SCHEMBL29634669

SCHEMBL29634669

COc1ccc(CNc2ncnc(Cl)c2N)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.58
EGFR P00533 3/20 0.56
KDM4C Q9H3R0 1/20 0.56
POLB P06746 1/20 0.56
NR2F2 P24468 1/20 0.56
GALR3 O60755 1/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
PDE5A O76074 1/20 0.54
LMNA P02545 2/20 0.54
MAPT P10636 2/20 0.54
TP53 P04637 1/20 0.54
RXFP1 Q9HBX9 1/20 0.54
ALDH1A1 P00352 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
THRB P10828 1/20 0.52
RAB9A P51151 1/20 0.51
CDK1 P06493 3/20 0.51
CCNB2 O95067 2/20 0.51
CCNB1 P14635 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233252 1.00 HTT (0.58) HTTEGFRKDM4CPOLBNR2F2
SCHEMBL11827284 0.83 STAT1 (0.62) HTTKDM4CPOLBGALR3MEN1
SCHEMBL16781105 0.82 LMNA (0.58) HTTEGFRPOLBNR2F2MEN1
SCHEMBL7746233 0.82 CNR1 (0.54) KDM4CGALR3MAPTALDH1A1RAB9A
SCHEMBL10873653 0.81 KDM4C (0.60) HTTEGFRKDM4CPOLBGALR3
SCHEMBL18786736 0.81 HTT (0.56) HTTEGFRPOLBNR2F2MEN1
SCHEMBL783719 0.81 KDM4C (0.72) HTTEGFRKDM4CNR2F2GALR3
SCHEMBL30983851 0.81 KDM4C (0.72) HTTEGFRKDM4CNR2F2GALR3
SCHEMBL20061544 0.81 AURKA (0.59) HTTEGFRPOLBNR2F2MEN1
SCHEMBL22307619 0.81 CYP1A2 (0.58) MEN1KMT2ALMNAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3514149-B1 HETEROCYCLIC AMIDE COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2022-05-18 EP disclosed